Cart
sales@molnova.com
Home - Products - Others - Other Targets - Acetyl-(Ala11·15)-Endothelin-1 (6-21)

Acetyl-(Ala11·15)-Endothelin-1 (6-21)

CAS No. 143113-45-5

Acetyl-(Ala11·15)-Endothelin-1 (6-21)( ——— )

Catalog No. M40168 CAS No. 143113-45-5

BQ-3020 is a selective endothelin receptor (ETB receptor) agonist that displaces [125I] ET-1 binding to ETB receptors, with an IC50 value of 0.2 nM. BQ-3020 elicits vasoconstriction in the rabbit pulmonary artery. BQ-3020 makes relaxation of the pig urinary bladder neck and can be used for cardiovascular disease research12.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
25MG Get Quote Get Quote
50MG Get Quote Get Quote
100MG Get Quote Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote
Get Quotation Bulk Inquiry Add to Cart

Biological Information

  • Product Name
    Acetyl-(Ala11·15)-Endothelin-1 (6-21)
  • Note
    Research use only, not for human use.
  • Brief Description
    BQ-3020 is a selective endothelin receptor (ETB receptor) agonist that displaces [125I] ET-1 binding to ETB receptors, with an IC50 value of 0.2 nM. BQ-3020 elicits vasoconstriction in the rabbit pulmonary artery. BQ-3020 makes relaxation of the pig urinary bladder neck and can be used for cardiovascular disease research12.
  • Description
    BQ-3020 is a selective endothelin receptor (ETB receptor) agonist that displaces [125I] ET-1 binding to ETB receptors, with an IC50 value of 0.2 nM.
  • In Vitro
    ———
  • In Vivo
    Animal Model:Cancer pain mouse model Dosage:3 mg/kg Administration:Injected subcutaneously at the site of the greatest tumor development Result:Attenuated cancer pain by approximately 50% up to 3 h post-injection compared to PBS-vehicle and contralateral injection
  • Synonyms
    ———
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    ETB: 0.2 nM (IC50)
  • Research Area
    ———
  • Indication
    ———

Chemical Information

  • CAS Number
    143113-45-5
  • Formula Weight
    1989.36
  • Molecular Formula
    C96H139N20O24S
  • Purity
    >98% (HPLC)
  • Solubility
    ———
  • SMILES
    ———
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Arteaga JL,et.al. Endothelin ET(B) receptors are involved in the relaxation to the pig urinary bladder neck. Neurourol Urodyn. 2012 Jun;31(5):688-94. ?
Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog
related products

  • Dehydrocorydalin

    Dehydrocorydaline exerts anti-metastatic potential via suppression of MMPs and Bcl-2 signaling in NSCLC cells.

  • 12-Hydroxyganodereni...

    12β-Hydroxyganoderenic acid B (Compound 15) is the triterpenoid compound that can be isolated from Ganoderma lucidum. Some triterpenoids isolated from Ganoderma species are reported to exhibits antitumor, antimicrobial, antiviral and anti-aging activities.

  • Vaccarin E

    Vaccarin E is a natural product of Vaccaria, Caryophyllaceae. Vaccarin E can be used as a reference standard.

Sign In Join Free