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Home - Products - Others - Other Targets - Acetyl-(Ala11·15)-Endothelin-1 (6-21)

Acetyl-(Ala11·15)-Endothelin-1 (6-21)

CAS No. 143113-45-5

Acetyl-(Ala11·15)-Endothelin-1 (6-21)( ——— )

Catalog No. M40168 CAS No. 143113-45-5

BQ-3020 is a selective endothelin receptor (ETB receptor) agonist that displaces [125I] ET-1 binding to ETB receptors, with an IC50 value of 0.2 nM. BQ-3020 elicits vasoconstriction in the rabbit pulmonary artery. BQ-3020 makes relaxation of the pig urinary bladder neck and can be used for cardiovascular disease research12.

Purity : >98% (HPLC)

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Biological Information

  • Product Name
    Acetyl-(Ala11·15)-Endothelin-1 (6-21)
  • Note
    Research use only, not for human use.
  • Brief Description
    BQ-3020 is a selective endothelin receptor (ETB receptor) agonist that displaces [125I] ET-1 binding to ETB receptors, with an IC50 value of 0.2 nM. BQ-3020 elicits vasoconstriction in the rabbit pulmonary artery. BQ-3020 makes relaxation of the pig urinary bladder neck and can be used for cardiovascular disease research12.
  • Description
    BQ-3020 is a selective endothelin receptor (ETB receptor) agonist that displaces [125I] ET-1 binding to ETB receptors, with an IC50 value of 0.2 nM.
  • In Vitro
    ———
  • In Vivo
    Animal Model:Cancer pain mouse model Dosage:3 mg/kg Administration:Injected subcutaneously at the site of the greatest tumor development Result:Attenuated cancer pain by approximately 50% up to 3 h post-injection compared to PBS-vehicle and contralateral injection
  • Synonyms
    ———
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    ETB: 0.2 nM (IC50)
  • Research Area
    ———
  • Indication
    ———

Chemical Information

  • CAS Number
    143113-45-5
  • Formula Weight
    1989.36
  • Molecular Formula
    C96H139N20O24S
  • Purity
    >98% (HPLC)
  • Solubility
    ———
  • SMILES
    ———
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Arteaga JL,et.al. Endothelin ET(B) receptors are involved in the relaxation to the pig urinary bladder neck. Neurourol Urodyn. 2012 Jun;31(5):688-94. ?
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