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LGD-2226
CAS No. 328947-93-9
LGD-2226( LGD2226 )
Catalog No. M14078 CAS No. 328947-93-9
LGD-2226 (LGD2226) is an orally active, selective androgen receptor modulator (SARM) with binding Ki of 1 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 873 | Get Quote |
|
| 50MG | 1782 | Get Quote |
|
| 100MG | 2250 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameLGD-2226
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NoteResearch use only, not for human use.
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Brief DescriptionLGD-2226 (LGD2226) is an orally active, selective androgen receptor modulator (SARM) with binding Ki of 1 nM.
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DescriptionLGD-2226 (LGD2226) is an orally active, selective androgen receptor modulator (SARM) with binding Ki of 1 nM, >1000-fold selectivity over GR,PR, MR and ER; LGD2226 is fully active in cell-based models of bone and muscle, exhibits anabolic activity on muscle and bone with reduced impact on prostate growth in rodent models; LGD2226 is also efficacious in a sex-behavior model in male rats measuring mounts, intromissions, ejaculations, and copulation efficiency.Osteoporosis Discontinued.
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In Vitro——
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In Vivo——
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SynonymsLGD2226
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PathwayEndocrinology/Hormones
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TargetAndrogen Receptor (AR)
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RecptorAndrogen Receptor (AR)
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Research AreaMetabolic Disease
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IndicationOsteoporosis
Chemical Information
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CAS Number328947-93-9
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Formula Weight392.225
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Molecular FormulaC14H9F9N2O
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C1NC2=C(C=C(N(CC(F)(F)F)CC(F)(F)F)C=C2)C(C(F)(F)F)=C1
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Chemical Name6-(bis-(2,2,2-trifluoroethyl)amino)-4-trifluoromethyl-1H-quinolin-2-one
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Miner JN, et al. Endocrinology. 2007 Jan;148(1):363-73.
2. van Oeveren A, et al. J Med Chem. 2006 Oct 19;49(21):6143-6.
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