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K00546
CAS No. 443798-47-8
K00546 ( K 00546 )
Catalog No. M14518 CAS No. 443798-47-8
K00546 is a potent inhibitor of the CDC2-like kinase CLK1 and CLK3 with IC50 of 8.9 and 29.2 nM, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 50MG | 1062 | Get Quote |
|
| 100MG | 1638 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameK00546
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NoteResearch use only, not for human use.
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Brief DescriptionK00546 is a potent inhibitor of the CDC2-like kinase CLK1 and CLK3 with IC50 of 8.9 and 29.2 nM, respectively.
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DescriptionK00546 is a potent inhibitor of the CDC2-like kinase CLK1 and CLK3 with IC50 of 8.9 and 29.2 nM, respectively.
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SynonymsK 00546
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PathwayCell Cycle/DNA Damage
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TargetCLK
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RecptorCLK
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Research Area——
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Indication——
Chemical Information
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CAS Number443798-47-8
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Formula Weight425.43
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Molecular FormulaC15H13F2N7O2S2
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Purity>98% (HPLC)
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Solubility——
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SMILESC1=CC(=C(C(=C1)F)NC(=S)N2C(=NC(=N2)NC3=CC=C(C=C3)S(=O)(=O)N)N)F
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Chemical Name5-amino-N-(2,6-difluorophenyl)-3-((4-sulfamoylphenyl)amino)-1H-1,2,4-triazole-1-carbothioamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Fedorov O, et al. Chem Biol. 2011 Jan 28;18(1):67-76.
2. Prak K, et al. Biochemistry. 2016 Jan 26;55(3):608-17.
2. Prak K, et al. Biochemistry. 2016 Jan 26;55(3):608-17.
molnova catalog
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K00546
K00546 is a potent inhibitor of the CDC2-like kinase CLK1 and CLK3 with IC50 of 8.9 and 29.2 nM, respectively.
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