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EPZ005687
CAS No. 1396772-26-1
EPZ005687 ( —— )
Catalog No. M11655 CAS No. 1396772-26-1
EPZ005687 is a potent and selective inhibitor of EZH2 with Ki of 24 nM in a cell-free assay.
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 48 | In Stock |
|
| 10MG | 69 | In Stock |
|
| 25MG | 124 | In Stock |
|
| 50MG | 186 | In Stock |
|
| 100MG | 332 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameEPZ005687
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NoteResearch use only, not for human use.
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Brief DescriptionEPZ005687 is a potent and selective inhibitor of EZH2 with Ki of 24 nM in a cell-free assay.
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DescriptionEPZ005687 is a potent and selective inhibitor of EZH2 with Ki of 24 nM in a cell-free assay, 50-fold selectivity against EZH1 and 500-fold selectivity against 15 other protein methyltransferases.
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Synonyms——
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PathwayChromatin/Epigenetic
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TargetHMTase
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RecptorEZH2
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1396772-26-1
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Formula Weight539.67
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Molecular FormulaC32H37N5O3
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Purity>98%(HPLC)
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SolubilityDMSO: 2 mg/mL (3.7 mM)
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SMILESCC1=CC(C)=C(CNC(=O)C2=C3C=NN(C4CCCC4)C3=CC(=C2)C2=CC=C(CN3CCOCC3)C=C2)C(=O)N1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Knutson SK, et al. Nat Chem Biol, 2012, 8(11), 890-896.
molnova catalog
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